Ex vivo and in vivo evaluation of (2R,3R)-5-[18F]-fluoroethoxy- and fluoropropoxy-benzovesamicol, as PET radioligands for the vesicular acetylcholine transporter-Reference-Cited by-同舟云学术

Ex vivo and in vivo evaluation of (2R,3R)-5-[18F]-fluoroethoxy- and fluoropropoxy-benzovesamicol, as PET radioligands for the vesicular acetylcholine transporter

Published:2007 Issue:12 Volume:61 Page:962-970
ISSN:0887-4476
Container-title:Synapse
language:en
Short-container-title:Synapse

Author:

Giboureau Nicolas,Emond Patrick,Fulton Roger R.,Henderson David J.,Chalon Sylvie,Garreau Lucette,Roselt Peter,Eberl Stefan,Mavel Sylvie,Bodard Sylvie,Fulham Michael J.,Guilloteau Denis,Kassiou Michael

Publisher

Wiley

Subject

Cellular and Molecular Neuroscience

Reference37 articles.

1. [3H]vesamicol binding in brain: Autoradiographic distribution, pharmacology, and effects of cholinergic lesions

2. Demonstration of a receptor in Torpedo synaptic vesicles for the acetylcholine storage blocker L-trans-2-(4-phenyl[3,4-3H]-piperidino) cyclohexanol.

3. A kinetic and allosteric model for the acetylcholine transporter-vesamicol receptor in synaptic vesicles

4. Piperazine analog of vesamicol: In vitro and in vivo characterization for vesicular acetylcholine transporter

5. Comparative metabolism of the designer drug 4-methylthioamphetamine by hepatocytes from man, monkey, dog, rabbit, rat and mouse

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