Rational truncation, mutation, and halogenation of bradykinin neuropeptides as potent ACEII inhibitors by integrating molecular dynamics simulations, quantum mechanics calculations, and in vitro assays
Author:
Affiliation:
1. Department of Neurology Suzhou Kowloon Hospital, Shanghai Jiao Tong University School of Medicine Suzhou China
2. Institute of Life Sciences Jiangsu University Zhenjiang China
Publisher
Wiley
Subject
General Chemistry
Link
https://onlinelibrary.wiley.com/doi/pdf/10.1002/jccs.202200242
Reference53 articles.
1. A Human Homolog of Angiotensin-converting Enzyme
2. Role of brain renin angiotensin system in neurodegeneration: An update
3. ACE2/ANG-(1–7)/Mas pathway in the brain: the axis of good
4. Brain-Selective Overexpression of Human Angiotensin-Converting Enzyme Type 2 Attenuates Neurogenic Hypertension
5. Angiotensin-converting enzyme 2 in the brain: properties and future directions
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