Identification of inactive conformation‐selective interleukin‐2‐inducible T‐cell kinase ( ITK ) inhibitors based on second‐harmonic generation-Reference-Cited by-同舟云学术

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Identification of inactive conformation‐selective interleukin‐2‐inducible T‐cell kinase ( ITK ) inhibitors based on second‐harmonic generation

Published:2018-07-30 Issue:9 Volume:8 Page:1412-1423
ISSN:2211-5463
Container-title:FEBS Open Bio
language:en
Short-container-title:FEBS Open Bio

Author:

Hantani Yoshiji¹,Iio Kiyosei²,Hantani Rie¹,Umetani Kayo¹,Sato Toshihiro¹,Young Tracy³,Connell Katelyn³,Kintz Sam³,Salafsky Joshua³

Affiliation:

1. Biological/Pharmacological Research Laboratories Central Pharmaceutical Research Institute Japan Tobacco Inc. Takatsuki Osaka Japan

2. Chemistry Research Laboratories Central Pharmaceutical Research Institute Japan Tobacco Inc. Takatsuki Osaka Japan

3. Biodesy, Inc. South San Francisco CA USA

Publisher

Wiley

Subject

General Biochemistry, Genetics and Molecular Biology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/2211-5463.12489

Reference33 articles.

1. The Protein Kinase Complement of the Human Genome

2. Protein kinases — the major drug targets of the twenty-first century?

3. Crystal Structure of the Catalytic Subunit of Cyclic Adenosine Monophosphate-Dependent Protein Kinase

4. Surface comparison of active and inactive protein kinases identifies a conserved activation mechanism

5. A quantitative analysis of kinase inhibitor selectivity

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. On the models for understanding the second harmonic generation scattering from lipid membranes and the corresponding molecular kinetics;Colloids and Surfaces A: Physicochemical and Engineering Aspects;2024-02

2. Conformational Selectivity of ITK Inhibitors: Insights from Molecular Dynamics Simulations;Journal of Chemical Information and Modeling;2023-12-09

3. Screening and biophysics in small molecule discovery;Small Molecule Drug Discovery;2020

4. Second-harmonic generation-based methods to detect and characterize ligand-induced RNA conformational changes;Methods;2019-09

5. Identification of a New Inhibitor That Stabilizes Interleukin-2-Inducible T-Cell Kinase in Its Inactive Conformation;SLAS DISCOVERY: Advancing the Science of Drug Discovery;2019-06-27

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