Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H3and H4Receptor Ligands
Author:
Affiliation:
1. Faculty of Chemistry and Pharmacy, Department of Pharmaceutical/Medicinal Chemistry II; University of Regensburg; Regensburg Germany
Publisher
Wiley
Subject
Drug Discovery,Pharmaceutical Science
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1002/ardp.201300316/fullpdf
Reference67 articles.
1. Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in Leukocytes
2. Molecular Cloning and Characterization of a New Human Histamine Receptor, HH4R
3. Discovery of a Novel Member of the Histamine Receptor Family
4. Cloning, Expression, and Pharmacological Characterization of a Novel Human Histamine Receptor
Cited by 14 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists;Journal of Medicinal Chemistry;2021-06-10
2. Discovery of a G Protein-Biased Radioligand for the Histamine H2 Receptor with Reversible Binding Properties;Journal of Medicinal Chemistry;2020-10-27
3. UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors;Journal of Medicinal Chemistry;2020-05-18
4. 4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H3 Receptor Agonists with in Vivo Central Nervous System Activity;Journal of Medicinal Chemistry;2019-11-01
5. [3H]UR-DEBa176: A 2,4-Diaminopyrimidine-Type Radioligand Enabling Binding Studies at the Human, Mouse, and Rat Histamine H4 Receptors;Journal of Medicinal Chemistry;2019-08-30
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3