Discovery and antiproliferative evaluation of new quinoxalines as potential DNA intercalators and topoisomerase II inhibitors

Author:

Eissa Ibrahim H.1ORCID,Metwaly Ahmed M.2,Belal Amany34ORCID,Mehany Ahmed B.M.5,Ayyad Rezk R.1,El‐Adl Khaled16ORCID,Mahdy Hazem A.1,Taghour Mohammed S.1,El‐Gamal Kamal M.A.7,El‐Sawah Mohamad E.7,Elmetwally Souad A.8,Elhendawy Mostafa. A.9,Radwan Mohamed M.910,ElSohly Mahmoud A.911

Affiliation:

1. Pharmaceutical Medicinal Chemistry Department, Faculty of Pharmacy (Boys) Al‐Azhar University Cairo Egypt

2. Department of Pharmacognosy, Faculty of Pharmacy (Boys) Al‐Azhar University Cairo Egypt

3. Department of Medicinal Chemistry, Faculty of Pharmacy Beni‐Suef University Beni‐Suef Egypt

4. Department of Pharmaceutical Chemistry, College of Pharmacy Taif University Taif Saudi Arabia

5. Department of Zoology, Faculty of Science Al‐Azhar University Cairo Egypt

6. Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Drug Technology Heliopolis University for Sustainable Development Cairo Egypt

7. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy (Boys) Al‐Azhar University Cairo Egypt

8. Department of Basic Science Higher Technological Institute 10th of Ramadan City Egypt

9. National Center for Natural Products Research University of Mississippi Mississippi

10. Department of Pharmacognosy, Faculty of Pharmacy Alexandria University Alexandria Egypt

11. Department of Pharmaceutics and Drug Delivery University of Mississippi Mississippi Mississippi

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Reference57 articles.

1. WHO Cancer Fact Sheet 2018 (accessed October 2018). Retrieved fromhttp://www.who.int/news‐room/fact‐sheets/detail/cancer.

2. Classification of anticancer drugs—a new system based on therapeutic targets

3. DNA and its associated processes as targets for cancer therapy

4. Cellular roles of DNA topoisomerases: a molecular perspective

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