Multiple Pathways Are Involved in the Oral Absorption of BMS-262084, a Tryptase Inhibitor, in Rats: Role of Paracellular Transport, Binding to Trypsin, and P-Glycoprotein Efflux-Reference-Cited by-同舟云学术

Multiple Pathways Are Involved in the Oral Absorption of BMS-262084, a Tryptase Inhibitor, in Rats: Role of Paracellular Transport, Binding to Trypsin, and P-Glycoprotein Efflux

Published:2005-05 Issue:5 Volume:94 Page:1115-1123
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Kamath Amrita V.,Morrison Richard A.,Harper Timothy W.,Lan Shih-Jung,Marino Anthony M.,Chong Saeho

Publisher

Elsevier BV

Subject

Pharmaceutical Science

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4. Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors;Sutton;Bioorg Med Chem Lett,2002

5. Uptake and transepithelial transport of the orally absorbed cephalosporin cephalexin, in the human intestinal cell line, Caco-2;Gochoco;Int J Pharm,1994

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