5-HT6antagonists as potential treatment for cognitive dysfunction

Author:

Liu Kevin G.,Robichaud Albert J.

Publisher

Wiley

Subject

Drug Discovery

Reference204 articles.

1. Interaction of chiral MS-245 analogs at h5-HT6 receptors;Abate;Bioorg Med Chem Lett,2005

2. Ahmed M, Johnson CN, Jones MC, MacDonald GJ, Moss SF, Thompson M, Wade CE, Witty D. 2003. Preparation of arylsulfonyl(diazacycloalkyl)quinolines for treatment of CNS disorders. WO Patent 2003080580.

3. Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists;Ahmed;Bioorg Med Chem Lett,2005

4. Ahmed M, Johnson CN, Miller ND, Trani G, Witty DR. 2005b. Preparation of 3-[(hetero)arylsulfonyl]-8-[(aminoalkyl)oxy]quinolines as 5-HT6 receptor antagonists for the treatment of CNS disorders. WO Patent 2005095346.

5. Beard CC, Clark RD, Fisher LE, Harris III RN, Repke DB. 2002. Preparation of new indole derivatives with 5-HT6 receptor affinity. WO Patent 2002098857.

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