The synthesis of one H-2 labeled and two H-3 labeled leukotriene C4 synthase inhibitors-Reference-Cited by-同舟云学术

The synthesis of one H-2 labeled and two H-3 labeled leukotriene C4 synthase inhibitors

Published:2020-07-07 Issue:10 Volume:63 Page:434-441
ISSN:0362-4803
Container-title:Journal of Labelled Compounds and Radiopharmaceuticals
language:en
Short-container-title:J Label Compd Radiopharm

Author:

Bergare Jonas¹,Kingston Lee¹^ORCID,Guly Dominic J.²,Dolan James²,Lewis Richard J.³^ORCID,Elmore Charles S.¹^ORCID

Affiliation:

1. Isotope Chemistry, Pharmaceutical Science, R&D; AstraZeneca; Gothenberg Sweden

2. Key Organics Ltd; Highfield Road Industrial Estate; Camelford PL32 9RA UK

3. Medicinal Chemistry, Research and Early Development, Respiratory, Inflammation and Autoimmune, BioPharmaceuticals R&D; AstraZeneca; Gothenberg Sweden

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Drug Discovery,Radiology, Nuclear Medicine and imaging,Biochemistry,Analytical Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/jlcr.3862/fullpdf

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4. Pharmacology of montelukast sodium (Singulair™), a potent and selective leukotriene D4 receptor antagonist;Jones;Can J Physiol Pharmacol,1995

5. Evolution of a series of peptidoleukotriene antagonists: synthesis and structure/activity relationships of 1,3,5-substituted indoles and indazoles;Matassa;J Med Chem,1990

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