Ritterostatin GN1N, a Cephalostatin-Ritterazine Bis-steroidal Pyrazine Hybrid, Selectively Targets GRP78

Author:

Ambrose Andrew J.1ORCID,Santos Evelyne A.2,Jimenez Paula C.23,Rocha Danilo D.2,Wilke Diego V.2,Beuzer Paolo4,Axelrod Josh4,Kumar Kanduluru Ananda56ORCID,Fuchs Philip L.5,Cang Hu4ORCID,Costa-Lotufo Letícia V.27ORCID,Chapman Eli1ORCID,La Clair James J.8ORCID

Affiliation:

1. Department of Pharmacology and Toxicology; College of Pharmacy; University of Arizona; 1703 East Mabel Street P. O. Box 210207 Tuscon AZ 85721 USA

2. Departamento de Fisiologia e Farmacologia; Universidade Federal do Ceará; Fortaleza CE 60.430-270 Brazil

3. Instituto do Mar; Universidade Federal de São Paulo; Santos SP 11.070-100 Brazil

4. Waitt Advanced Biophotonics Center; The Salk Institute for Biological Sciences; 10010 North Torrey Pines Road La Jolla CA 92037 USA

5. Department of Chemistry; Purdue University; West Lafayette IN 47907 USA

6. Present address: On Target Laboratories; 1281 Win Hentschel Boulevard West Lafayette IN 47907 USA

7. Departamento de Farmacologia; Universidade de São Paulo; São Paulo SP 05508-900 Brazil

8. Xenobe Research Institute; P. O. Box 3052 San Diego CA 92163-1052 USA

Publisher

Wiley

Subject

Organic Chemistry,Molecular Biology,Molecular Medicine,Biochemistry

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