Chemoselective Preparation of Clickable Aryl Sulfonyl Fluoride Monomers: A Toolbox of Highly Functionalized Intermediates for Chemical Biology Probe Synthesis
Author:
Affiliation:
1. Medicine Design; Pfizer Inc.; Eastern Point Road Groton CT 06340 USA
2. Oncology RU Medicinal Chemistry; Pfizer Inc.; 10770 Science Center Drive San Diego CA 92121 USA
3. Medicine Design; Pfizer Inc.; 610 Main Street Cambridge MA 02139 USA
Publisher
Wiley
Subject
Organic Chemistry,Molecular Biology,Molecular Medicine,Biochemistry
Reference24 articles.
1. Sulfonyl fluorides as privileged warheads in chemical biology
2. Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry
3. Schwefel(VI)-fluorid-Austausch (SuFEx): Eine weitere gute Anwendung für die Click-Chemie
4. Spontaneous hydrolysis of sulfonyl fluorides
5. Selective Targeting of Distinct Active Site Nucleophiles by Irreversible Src-Family Kinase Inhibitors
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