HDAC4 Inhibitors with Cyclic Linker and Non‐hydroxamate Zinc Binding Group: Design, Synthesis, HDAC Screening and in vitro Cytotoxicity evaluation.-Reference-Cited by-同舟云学术

HDAC4 Inhibitors with Cyclic Linker and Non‐hydroxamate Zinc Binding Group: Design, Synthesis, HDAC Screening and in vitro Cytotoxicity evaluation.

Published:2021-07-12 Issue:26 Volume:6 Page:6748-6763
ISSN:2365-6549
Container-title:ChemistrySelect
language:en
Short-container-title:ChemistrySelect

Author:

Tilekar Kalpana¹,Hess Jessica D.²,Upadhyay Neha¹,Schweipert Markus³,Flath Felix³,Gutierrez Denisse A.²,Loiodice Fulvio⁴,Lavecchia Antonio⁵,Meyer‐Almes Franz‐Josef³,Aguilera Renato J.²,Ramaa C. S.¹

Affiliation:

1. Department of Pharmaceutical Chemistry Bharati Vidyapeeth's College of Pharmacy, Sector 8, CBD Belapur Navi Mumbai India

2. Cellular Characterization and Biorepository Core Facility Border Biomedical Research Center Department of Biological Sciences The University of Texas at El Paso 500 West University Avenue El Paso TX 79968-0519 USA

3. Department of Chemical Engineering and Biotechnology University of Applied Science Haardtring 100 64295 Darmstadt Germany

4. Department of Pharmacy-Drug Science University of Bari “Aldo Moro” Via E. Orabona, 4 70126 Bari Italy

5. Department of Pharmacy “Drug Discovery” Laboratory University of Napoli “Federico II” Via D. Montesano, 49 80131 Napoli Italy

Publisher

Wiley

Subject

General Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/slct.202102061

Reference65 articles.

1. Erasers of Histone Acetylation: The Histone Deacetylase Enzymes

2. Distribution of histone deacetylases 1–11 in the rat brain