Classifying protein kinase structures guides use of ligand-selectivity profiles to predict inactive conformations: Structure of lck/imatinib complex-Reference-Cited by-同舟云学术

Classifying protein kinase structures guides use of ligand-selectivity profiles to predict inactive conformations: Structure of lck/imatinib complex

Published:2007-10-01 Issue:4 Volume:70 Page:1451-1460
ISSN:0887-3585
Container-title:Proteins: Structure, Function, and Bioinformatics
language:en
Short-container-title:Proteins

Author:

Jacobs Marc D.,Caron Paul R.,Hare Brian J.

Publisher

Wiley

Subject

Molecular Biology,Biochemistry,Structural Biology

Reference42 articles.

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4. Crystal structures of the kinase domain of c-Abl in complex with the small molecule inhibitors PD173955 and imatinib (STI-571);Nagar;Cancer Res,2002

5. Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel noncompetitive kinase inhibition;Ohren;Nat Struct Mol Biol,2004

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