An Efficient One-Pot Synthesis of Chiral N-Protected 3-Substituted (Diketo)piperazines via Ugi-4CR/De-Boc/Cyclization Process-Reference-Cited by-同舟云学术

An Efficient One-Pot Synthesis of Chiral N-Protected 3-Substituted (Diketo)piperazines via Ugi-4CR/De-Boc/Cyclization Process

Published:2018-01-25 Issue:4 Volume:3 Page:1027-1031
ISSN:2365-6549
Container-title:ChemistrySelect
language:en
Short-container-title:ChemistrySelect

Author:

Jida Mouhamad¹,Ballet Steven¹

Affiliation:

1. Research Group of Organic Chemistry; Departments of Chemistry and Bioengineering Sciences; Vrije Universiteit Brussel; Pleinlaan 2 B-1050 Brussels Belgium

Funder

Vrije Universiteit Brussel

Publisher

Wiley

Subject

General Chemistry

Reference80 articles.

1. Structure-Based Exploration of Cyclic Dipeptide Chitinase Inhibitors

2. NPI-2358 is a tubulin-depolymerizing agent: in-vitro evidence for activity as a tumor vascular-disrupting agent

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Application of post-Ugi transformation strategies towards the synthesis and functionalization of 2,5-Diketopiperazines;Tetrahedron;2024-07

2. Curation and cheminformatics analysis of a Ugi-reaction derived library (URDL) of synthetically tractable small molecules for virtual screening application;Molecular Diversity;2022-12-27

3. Diketopiperazines as Chiral Building Blocks;Chiral Building Blocks in Asymmetric Synthesis;2022-08-12

4. One-Pot Diastereoselective Synthesis of Pyrrolopiperazine-2,6-diones by a Ugi/Nucleophilic Substitution/N-Acylation Sequence;The Journal of Organic Chemistry;2022-06-27

5. 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity;European Journal of Medicinal Chemistry;2022-01