Synthesis of Constrained Heterocycles Employing Two Post-Ugi Cyclization Methods for Rapid Library Generation with In Cellulo Activity-Reference-Cited by-同舟云学术

Synthesis of Constrained Heterocycles Employing Two Post-Ugi Cyclization Methods for Rapid Library Generation with In Cellulo Activity

Published:2017-12-11 Issue:35 Volume:2 Page:11821-11825
ISSN:2365-6549
Container-title:ChemistrySelect
language:en
Short-container-title:ChemistrySelect

Author:

McConnell Nicholas¹,Xu Zhigang²,Kumarasamy Vishnu¹,Sun Daekyu¹,Frett Brendan³,Li Hong-yu³

Affiliation:

1. Department of Pharmacology and Toxicology; University of Arizona; Tucson, Arizona 85719 United States

2. International Academy of Targeted Therapeutics and Innovation; Chongqing University of Arts and Sciences; 319 Honghe Ave., Yongchuan, Chongqing 402160 China

3. Department of Pharmaceutical Sciences; College of Pharmacy; University of Arkansas for Medical Sciences; Little Rock, Arkansas 72205 United States

Funder

National Institutes of Health

Publisher

Wiley

Subject

General Chemistry

Reference73 articles.

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2. Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent Polypharmacology

3. 4-(Aminoalkylamino)-3-benzimidazole-quinolinones as potent CHK-1 inhibitors

4. Green route for the heterocyclization of 2-mercaptobenzimidazole into β-lactum segment derivatives containing –CONH– bridge with benzimidazole: Screening in vitro antimicrobial activity with various microorganisms

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