Structure‐Enabled Discovery of a Stapled Peptide Inhibitor to Target the Oncogenic Transcriptional Repressor TLE1-Reference-Cited by-同舟云学术

Structure‐Enabled Discovery of a Stapled Peptide Inhibitor to Target the Oncogenic Transcriptional Repressor TLE1

Published:2017-06-27 Issue:40 Volume:23 Page:9577-9584
ISSN:0947-6539
Container-title:Chemistry – A European Journal
language:en
Short-container-title:Chem. Eur. J.

Author:

McGrath Sally¹,Tortorici Marcello¹,Drouin Ludovic¹,Solanki Savade¹,Vidler Lewis¹,Westwood Isaac¹,Gimeson Peter²,Van Montfort Rob³,Hoelder Swen¹

Affiliation:

1. The Institute of Cancer ResearchDivision of Cancer Therapeutics UnitCancer Research UK Cancer Therapeutics Unit 15 Cotswold Road, Sutton Surrey SM2 5NG UK

2. Malvern Instruments Nordic AB Vallongatan 1 Uppsala 752 28 Sweden

3. Cancer Research (UK) Cancer Therapeutics UnitDivision of Cancer TherapeuticsDivision of Structural BiologyThe Institute of Cancer Research 15 Cotswold Road, Sutton Surrey SM2 5NG UK

Funder

Wellcome Trust

Cancer Research UK

Publisher

Wiley

Subject

General Chemistry,Catalysis,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/chem.201700747

Reference25 articles.

2. The Groucho/TLE/Grg family of transcriptional co-repressors

3. Groucho/TLE family proteins and transcriptional repression

5. Immunohistochemical Staining for TLE1 Distinguishes Synovial Sarcoma From Histologic Mimics

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