Highly Efficient Synthesis of a Staphylococcus aureus Targeting Payload to Enable the First Antibody-Antibiotic Conjugate-Reference-Cited by-同舟云学术

Highly Efficient Synthesis of a Staphylococcus aureus Targeting Payload to Enable the First Antibody-Antibiotic Conjugate

Published:2017-12-08 Issue:12 Volume:24 Page:2837-2840
ISSN:0947-6539
Container-title:Chemistry - A European Journal
language:en
Short-container-title:Chem. Eur. J.

Author:

Linghu Xin¹,Segraves Nathaniel L.²,Abramovich Ifat²,Wong Nicholas¹,Müller Barbara¹,Neubauer Nadja¹,Fantasia Serena³,Rieth Sebastian³,Bachmann Stephan³,Jansen Michael³,Sowell C. Gregory¹,Askin David¹,Koenig Stefan G.¹^ORCID,Gosselin Francis¹

Affiliation:

1. Department of Small Molecule Process Chemistry; Genentech, Inc.; 1 DNA Way South San Francisco, CA 94080 USA

2. Department of Small Molecule Analytical Chemistry and Quality Control; Genentech, Inc.; 1 DNA Way South San Francisco, CA 94080 USA

3. Pharma Technical Development, Process Chemistry & Catalysis; F. Hoffmann-La Roche Ltd.; Grenzacherstrasse 124 4070 Basel Switzerland

Publisher

Wiley

Subject

General Chemistry,Catalysis,Organic Chemistry

Reference46 articles.

1. How to cope with the quest for new antibiotics

2. Introduction to Antibiotic Resistance

3. The Evolving Role of Chemical Synthesis in Antibacterial Drug Discovery

4. Zur Rolle der chemischen Synthese in der Entwicklung antibakterieller Wirkstoffe

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