Drug Syntheses Beyond the Rule of 5
Author:
Affiliation:
1. Department of Chemistry–BMC Uppsala University Box 576 75123 Uppsala Sweden
2. Department of Medicinal Chemistry, MIPS Monash University 381 Royal Parade Parkville Victoria 3052 Australia
Funder
Vetenskapsrådet
Publisher
Wiley
Subject
General Chemistry,Catalysis,Organic Chemistry
Link
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chem.201902716
Reference181 articles.
1. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
2. Structural Biology and Drug Discovery of Difficult Targets: The Limits of Ligandability
3. Oral Druggable Space beyond the Rule of 5: Insights from Drugs and Clinical Candidates
4. How proteins bind macrocycles
5. How Beyond Rule of 5 Drugs and Clinical Candidates Bind to Their Targets
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