Discovery of a novel fluorescent chemical probe suitable for evaluation of neuropilin‐1 binding of small molecules-Reference-Cited by-同舟云学术

Discovery of a novel fluorescent chemical probe suitable for evaluation of neuropilin‐1 binding of small molecules

Published:2020-01-20 Issue:4 Volume:81 Page:491-500
ISSN:0272-4391
Container-title:Drug Development Research
language:en
Short-container-title:Drug Dev Res

Author:

Conole Daniel¹,Chou Yi‐Tai¹,Patsiarika Anastasia¹,Nwabo Valery¹,Dimitriou Eleni¹,Soudy Christelle¹,Mota Filipa¹,Djordjevic Snezana²,Selwood David L.¹^ORCID

Affiliation:

1. Wolfson Institute for Biomedical ResearchUniversity College London London UK

2. Institute of Structural and Molecular BiologyUniversity College London London UK

Funder

British Heart Foundation

Publisher

Wiley

Subject

Drug Discovery

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ddr.21641

Reference22 articles.

1. Gain of affinity for VEGF165 binding within the VEGFR2/NRP1 cellular complex detected by an HTRF-based binding assay

2. IC50-to-Ki: a web-based tool for converting IC50 to Ki values for inhibitors of enzyme activity and ligand binding

3. Stability and function of regulatory T cells is maintained by a neuropilin-1–semaphorin-4a axis

4. Fluorescence polarization assay to quantify protein‐protein interactions in an HTS format;Du Y. H.;Protein‐Protein Interactions: Methods and Applications, 2nd Edition,2015

5. VEGF-A acts via neuropilin-1 to enhance epidermal cancer stem cell survival and formation of aggressive and highly vascularized tumors

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