Method development and validation for simultaneous determination of ebastine and its active metabolite carebastine in human plasma by liquid chromatography–tandem mass spectrometry and its application to a clinical pharmacokinetic study in healthy Chinese volunteers

Author:

Phiri Margaret12ORCID,Li Duo1,Li Tengfei1,Ji Shunli1,Ling Tang12,Li Xianjing12,Gao Huaye12,Ding Li12ORCID,Shu Chang1

Affiliation:

1. Department of Pharmaceutical Analysis China Pharmaceutical University 639 Longmian avenue, jiangning Nanjing jiangsu China

2. Nanjing Clinical Tech Laboratories Inc. Nanjing China

Funder

National Natural Science Foundation of China

Publisher

Wiley

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,General Medicine,Biochemistry,Analytical Chemistry

Reference24 articles.

1. Idiopathic Chronic Urticaria and Celiac Disease

2. Comparative Efficacy and Safety of Ebastine 20 mg, Ebastine 10 mg and Levocetirizine 5 mg in Acute Urticaria;Goyal V.;Journal of Clinical and Diagnostic Research,2017

3. Chronic idiopathic urticaria

4. Involvement of CYP2J2 and CYP4F12 in the Metabolism of Ebastine in Human Intestinal Microsomes

5. Pharmacokinetics and Electrocardiographic Effect of Ebastine in Young Versus Elderly Healthy Subjects

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