Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αV β3 -Integrin Ligands for Tumor Targeting-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αV β3 -Integrin Ligands for Tumor Targeting

Published:2018-06-01 Issue:23 Volume:2018 Page:2902-2909
ISSN:1434-193X
Container-title:European Journal of Organic Chemistry
language:en
Short-container-title:Eur. J. Org. Chem.

Author:

López Rivas Paula¹^ORCID,Ranđelović Ivan²^ORCID,Raposo Moreira Dias André¹^ORCID,Pina Arianna¹^ORCID,Arosio Daniela³^ORCID,Tóvári József²^ORCID,Mező Gábor⁴^ORCID,Dal Corso Alberto¹,Pignataro Luca¹^ORCID,Gennari Cesare¹³^ORCID

Affiliation:

1. Dipartimento di Chimica; Università degli Studi di Milano; Via C. Golgi, 19 20133 Milan Italy

2. Department of Experimental Pharmacology; National Institute of Oncology; Ráth György u. 7-9. 1122 Budapest Hungary

3. CNR; Istituto di Scienze e Tecnologie Molecolari (ISTM); Via C. Golgi, 19 20133 Milan Italy

4. Faculty of Science; Institute of Chemistry; Eötvös Loránd University; Pázmány Péter st. 1/A 1117 Budapest Hungary

Funder

Horizon 2020 Framework Programme

Ministero dell’Istruzione, dell’Università e della Ricerca

Publisher

Wiley

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/ejoc.201800447/fullpdf

Reference53 articles.

1. Antibody-Drug Conjugates: An Emerging Concept in Cancer Therapy

2. Antikörper-Wirkstoff-Konjugate: ein neues Konzept in der Krebstherapie

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5. Small Targeted Cytotoxics: Current State and Promises from DNA-Encoded Chemical Libraries

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