Structures of human Bruton's tyrosine kinase in active and inactive conformations suggest a mechanism of activation for TEC family kinases-Reference-Cited by-同舟云学术

Structures of human Bruton's tyrosine kinase in active and inactive conformations suggest a mechanism of activation for TEC family kinases

Published:2010-01-05 Issue:3 Volume:19 Page:429-439
ISSN:0961-8368
Container-title:Protein Science
language:en
Short-container-title:Protein Science

Author:

Marcotte Douglas J.,Liu Yu-Ting,Arduini Robert M.,Hession Catherine A.,Miatkowski Konrad,Wildes Craig P.,Cullen Patrick F.,Hong Victor,Hopkins Brian T.,Mertsching Elisabeth,Jenkins Tracy J.,Romanowski Michael J.,Baker Darren P.,Silvian Laura F.

Publisher

Wiley

Subject

Molecular Biology,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/pro.321/fullpdf

Reference30 articles.

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3. The gene involved in X-linked agammaglobulinaemia is a member of the src family of protein-tyrosine kinases;Vetrie;Nature,1993

4. Rational design and synthesis of a novel anti-leukemic agent targeting Bruton's tyrosine kinase (BTK), LFM-A13 [alpha-cyano-beta-hydroxy-beta-methyl-N-(2,5-dibromophenyl)propenamide];Mahajan;J Biol Chem,1999

5. The Btk inhibitor LFM-A13 is a potent inhibitor of Jak2 kinase activity;van den Akker;Biol Chem,2004

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