Integrating Dynamic Positron Emission Tomography and Conventional Pharmacokinetic Studies to Delineate Plasma and Tumor Pharmacokinetics of FAU, a Prodrug Bioactivated by Thymidylate Synthase
Author:
Affiliation:
1. Karmanos Cancer Institute; Department of Oncology; Wayne State University School of Medicine; Detroit MI USA
2. Department of Radiology; Wayne State University; Detroit MI USA
3. Yale Cancer Center; Yale School of Medicine; New Haven CT USA
Funder
United States Public Health
Service Cancer Center
National Institutes of Health
Publisher
Wiley
Subject
Pharmacology (medical),Pharmacology
Reference39 articles.
1. Positron emission tomography and drug discovery: contributions to the understanding of pharmacokinetics, mechanism of action and disease state characterization;Klimas;Mol Imag Biol,2002
2. Application of PET/CT in the development of novel anticancer drugs;Boss;Oncologist,2008
3. Plasma pharmacokinetic evaluation of cytotoxic agents radiolabelled with positron emitting radioisotopes;Saleem;Cancer Chemother Pharmacol,2008
4. Pharmacokinetic analysis of 5-[18F]fluorouracil tissue concentrations measured with positron emission tomography in patients with liver metastases from colorectal adenocarcinoma;Kissel;Cancer Res,1997
5. Distribution of 1-(2-deoxy-2-fluoro-beta-D-arabinofuranosyl) uracil in mice bearing colorectal cancer xenografts: rationale for therapeutic use and as a positron emission tomography probe for thymidylate synthase;Eiseman;Clin Cancer Res,2004
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