Differential Selectivity of Efflux Transporter Inhibitors in Caco-2 and MDCK–MDR1 Monolayers: A Strategy to Assess the Interaction of a New Chemical Entity with P-gp, BCRP, and MRP2-Reference-Cited by-同舟云学术

Differential Selectivity of Efflux Transporter Inhibitors in Caco-2 and MDCK–MDR1 Monolayers: A Strategy to Assess the Interaction of a New Chemical Entity with P-gp, BCRP, and MRP2

Published:2012-05 Issue:5 Volume:101 Page:1888-1897
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Mease Kirsten,Sane Rucha,Podila Lalitha,Taub Mitchell E.

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference47 articles.

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5. cDNA cloning of the hepatocyte canalicular isoform of the multidrug resistance protein, cMrp, reveals a novel conjugate export pump deficient in hyperbilirubinemic mutant rats;Büchler;J Biol Chem,1996

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