3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists-Reference-Cited by-同舟云学术

3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists

Published:2022-11-03 Issue:1 Volume:356 Page:2200432
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Archiv der Pharmazie

Author:

Tocco Graziella¹^ORCID,Laus Antonio¹,Vanejevs Maksims²,Ture Anastasija²,Mostallino Rafaela³,Pintori Nicholas³,De Luca Maria Antonietta³^ORCID,Castelli M. Paola³^ORCID,Di Chiara Gaetano³⁴

Affiliation:

1. Department of Life and Environmental Sciences, University of Cagliari Cittadella Universitaria di Monserrato, Monserrato Cagliari Italy

2. Laboratory of CNS Active Compounds Latvian Institute of Organic Chemistry Riga Latvia

3. Department of Biomedical Sciences, University of Cagliari Cittadella Universitaria di Monserrato, Monserrato Cagliari Italy

4. Neuroscience Institute National Research Council of Italy (CNR) Cagliari Italy

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ardp.202200432

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1. Propionamide Derivatives as Dual μ-Opioid Receptor Agonists and σ1 Receptor Antagonists for the Treatment of Pain

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3. Structure-activity relationships of trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidine antagonists for .mu.- and .kappa.-opioid receptors

4. The Discovery and Development of theN-Substitutedtrans-3,4-Dimethyl-4-(3′-hydroxyphenyl)piperidine Class of Pure Opioid Receptor Antagonists

5. 1-Substituted 4-(3-Hydroxyphenyl)piperazines Are Pure Opioid Receptor Antagonists

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