Triazoloquinazoline derived classical DNA intercalators: Design, synthesis, in silico ADME profile, docking, and antiproliferative evaluations
Author:
Affiliation:
1. Pharmaceutical Medicinal Chemistry and Drug Design Department Al‐Azhar University Cairo Egypt
2. Pharmaceutical Chemistry Department Heliopolis University for Sustainable Development Cairo Egypt
Publisher
Wiley
Subject
Drug Discovery,Pharmaceutical Science
Link
https://onlinelibrary.wiley.com/doi/pdf/10.1002/ardp.202100506
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3. Synthesis of [1,2,4]triazolo[4,3-a]quinoxaline-1,3,4-oxadiazole derivatives as potent antiproliferative agents via a hybrid pharmacophore approach
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5. Pyrimidoquinazoline-Based Antitumor Agents. Design of Topoisomerase II to DNA Cross-linkers with Activity against Protein Kinases
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