Structure‐based design, synthesis, and evaluation of Bcl‐2/Mcl‐1 dual inhibitors-Reference-Cited by-同舟云学术

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Structure‐based design, synthesis, and evaluation of Bcl‐2/Mcl‐1 dual inhibitors

Published:2020-03-16 Issue:5 Volume:353 Page:
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Arch Pharm

Author:

Zhu Junjie¹^ORCID,Wang Ziqian²,Guo Zongwei³,Zhang Xiaodong¹,Song Ting¹,Guo Yafei³,Ji Tong¹,Zhang Zhichao¹

Affiliation:

1. State Key Laboratory of Fine Chemicals, School of ChemistryDalian University of TechnologyDalian China

2. Zhang Dayu School of ChemistryDalian University of TechnologyDalian China

3. School of Life Science and TechnologyDalian University of TechnologyDalian China

Funder

National Natural Science Foundation of China

China Postdoctoral Science Foundation

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ardp.202000005

Reference32 articles.

1. Dual inhibitors of the pro-survival proteins Bcl-2 and Mcl-1 derived from natural compound meiogynin A

2. Deciphering the rules of programmed cell death to improve therapy of cancer and other diseases

3. Control of apoptosis by the BCL-2 protein family: implications for physiology and therapy

4. Design, synthesis and preliminary bioactivity studies of indomethacin derivatives as Bcl-2/Mcl-1 dual inhibitors

5. Combining BH3-mimetics to target both BCL-2 and MCL1 has potent activity in pre-clinical models of acute myeloid leukemia

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1. Design of Tracers in Fluorescence Polarization Assay for Extensive Application in Small Molecule Drug Discovery;Journal of Medicinal Chemistry;2023-08-10

2. Mixture-Based Screening of Focused Combinatorial Libraries by NMR: Application to the Antiapoptotic Protein hMcl-1;Journal of Medicinal Chemistry;2023-07-19

3. Identification of bicyclic compounds that act as dual inhibitors of Bcl-2 and Mcl-1;Molecular Diversity;2022-07-31

4. Structure-Based Design and Structure-Activity Relationship Analysis of Small Molecules Inhibiting Bcl-2 Family Members;Pharmaceutical Chemistry Journal;2022-05-28

5. Myeloid cell leukemia 1 (MCL-1): Structural characteristics and application in cancer therapy;International Journal of Biological Macromolecules;2021-09

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