Radiosynthesis of the 11 C-methyl derivative of LBQ657 for PET investigation of the neprilysin inhibitor sacubitril-Reference-Cited by-同舟云学术

Radiosynthesis of the 11 C-methyl derivative of LBQ657 for PET investigation of the neprilysin inhibitor sacubitril

Published:2020-01-08 Issue:2 Volume:63 Page:65-71
ISSN:0362-4803
Container-title:Journal of Labelled Compounds and Radiopharmaceuticals
language:en
Short-container-title:J Label Compd Radiopharm

Author:

Teyssier Valentin R.¹²,Simard José-Mathieu¹,Dornan Mark H.¹³,Tournoux François⁴⁵,DaSilva Jean N.¹²³^ORCID

Affiliation:

1. Laboratoire de Radiochimie et Cyclotron, Centre de Recherche du Centre Hospitalier de l'Université de Montréal, Montréal; Québec Canada

2. Institut de Génie Biomédical, Faculté de Médecine; Université de Montréal; Québec Canada

3. Département de Radiologie, radio-oncologie et médecine nucléaire, Faculté de médecine; Université de Montréal; Québec Canada

4. Département de Médecine, Centre de Recherche du Centre Hospitalier de l'Université de Montréal, Montréal; Québec Canada

5. Centre cardiovasculaire, Centre Hospitalier de l'Université de Montréal, Montréal; Québec Canada

Funder

Réseau en Bio-Imagerie du Quebec

SQIC-Roche

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Drug Discovery,Radiology, Nuclear Medicine and imaging,Biochemistry,Analytical Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/jlcr.3817/fullpdf

Reference19 articles.

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2. Novel O-[11C]-methylated derivatives of the neprilysin inhibitor sacubitril: Radiosynthesis, autoradiography and plasma stability evaluation;Nuclear Medicine and Biology;2021-11