Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione-Reference-Cited by-同舟云学术

Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione

Published:2015-03-13 Issue:4 Volume:348 Page:229-241
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Arch. Pharm. Chem. Life Sci.

Author:

Żmudzki Paweł¹,Chłoń-Rzepa Grażyna¹,Bojarski Andrzej J.²,Zygmunt Małgorzata³,Kazek Grzegorz⁴,Mordyl Barbara⁵,Pawłowski Maciej¹

Affiliation:

1. Department of Medicinal Chemistry; Jagiellonian University Medical College; Kraków Poland

2. Department of Medicinal Chemistry; Institute of Pharmacology; Polish Academy of Sciences; Kraków Poland

3. Department of Pharmacodynamics; Jagiellonian University Medical College; Kraków Poland

4. Department of Pharmacological Screening; Jagiellonian University Medical College; Kraków Poland

5. Department of Pharmacobiology; Jagiellonian University Medical College; Kraków Poland

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/ardp.201400392/fullpdf

Reference6 articles.

1. 7-Arylpiperazinylalkyl and 7-tetrahydroisoquinolinylalkyl derivatives of 8-alkoxy-purine-2,6-dione and some of their purine-2,6,8-trione analogs as 5-HT1A, 5-HT2A, and 5-HT7 serotonin receptor ligands

2. Patent Laboratoire Lebrun S.A. Pharmacologically Active 8-Aminotheophylline Derivatives 1972

3. M. Pawłowski Dissertation 1992 Akademia Medyczna im. M. Kopernika Cracow

4. Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT1A/5-HT2A/5-HT7 and dopamine D2/D3 receptors

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