Evaluation of Proposed In Vivo Probe Substrates and Inhibitors for Phenotyping Transporter Activity in Humans

Author:

Momper Jeremiah D.1,Tsunoda Shirley M.1,Ma Joseph D.1

Affiliation:

1. University of California, San Diego; Skaggs School of Pharmacy & Pharmaceutical Sciences; La Jolla CA USA

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Reference162 articles.

1. Membrane transporters in drug development;Giacomini;Nat Rev Drug Discov,2010

2. Emerging transporters of clinical importance: an update from the International Transporter Consortium;Hillgren;Clin Pharmacol Ther,2013

3. EMA. European Medicines Agency http://www.ema.europa.eu/docs/en_GB/document_library/Scientific_guideline/2012/07/WC500129606.pdf

4. FDA. Guidance for Industry http://www.fda.gov/downloads/drugs/guidancecomplianceregulatoryinformation/guidances/ucm292362.pdf

5. The UCSF-FDA TransPortal: a public drug transporter database;Morrissey;Clin Pharmacol Ther,2012

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