Initial Testing (Stage 1) of MK-8242-A Novel MDM2 Inhibitor-by the Pediatric Preclinical Testing Program

Author:

Kang Min H.1,Reynolds C. Patrick1,Kolb E. Anders2,Gorlick Richard3,Carol Hernan4,Lock Richard4,Keir Stephen T.5,Maris John M.6,Wu Jianwrong7,Lyalin Dmitry8,Kurmasheva Raushan T.8,Houghton Peter J.8,Smith Malcolm A.9

Affiliation:

1. Cancer Center; Texas Tech University Health Sciences Center; Lubbock Texas

2. A.I. duPont Hospital for Children; Wilmington Delaware

3. The Children's Hospital at Montefiore; Bronx New York

4. Children's Cancer Institute Australia for Medical Research; Randwick NSW Australia

5. Duke University Medical Center; Durham North Carolina

6. Children's Hospital of Philadelphia; University of Pennsylvania School of Medicine and Abramson Family Cancer Research Institute; Philadelphia Pennsylvania

7. St. Jude Children's Research Hospital; Memphis Tennessee

8. Nationwide Children's Hospital; Columbus Ohio

9. Cancer Therapy Evaluation Program; NCI; Bethesda Maryland

Funder

National Cancer Institute

Publisher

Wiley

Subject

Oncology,Hematology,Pediatrics, Perinatology and Child Health

Reference41 articles.

1. p53 in health and disease;Vousden;Nat Rev Mol Cell Biol,2007

2. p53 the cellular gatekeeper for growth and division;Levine;Cell,1997

3. p53 and disease: When the guardian angel fails;Royds;Cell Death Differ,2006

4. The relationship between TP53 mutations and overexpression of p53 and prognosis in malignant gliomas of childhood;Pollack;Cancer Res,1997

5. The p53 pathway and its inactivation in neuroblastoma;Tweddle;Cancer Lett,2003

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