Toward the design of cannabinoid CB1 receptor inverse agonists and neutral antagonists
Author:
Publisher
Wiley
Subject
Drug Discovery
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1002/ddr.20337/fullpdf
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3. Activation of the β2 adrenergic receptor involves disruption of an ionic link between the cytoplasmic ends of transmembrane segments 3 and 6;Ballesteros;J Biol Chem,2001
4. Agonist alkyl tail interaction with cannabinoid CB1 receptor V6.43/I6.46 groove induces a Helix 6 active conformation;Barnett-Norris;Int J Quantum Chem,2002
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