Design and Synthesis of Imidazole and Triazole Pyrazoles as Mycobacterium Tuberculosis CYP121A1 Inhibitors-Reference-Cited by-同舟云学术

Design and Synthesis of Imidazole and Triazole Pyrazoles as Mycobacterium Tuberculosis CYP121A1 Inhibitors

Published:2019-07 Issue:7 Volume:8 Page:995-1011
ISSN:2191-1363
Container-title:ChemistryOpen
language:en
Short-container-title:ChemistryOpen

Author:

Kishk Safaa M.¹²,McLean Kirsty J.³,Sood Sakshi⁴,Smith Darren¹,Evans Jack W.D.¹,Helal Mohamed A.²⁵,Gomaa Mohamed S.²⁶,Salama Ismail²,Mostafa Samia M.²,de Carvalho Luiz Pedro S.⁴,Levy Colin W.³,Munro Andrew W.³,Simons Claire¹^ORCID

Affiliation:

1. School of Pharmacy & Pharmaceutical SciencesCardiff University King Edward VII Avenue Cardiff CF10 3NB U.K.

2. Medicinal Chemistry Department, Faculty of PharmacySuez Canal University Ismailia Egypt

3. Manchester Institute of Biotechnology, School of ChemistryUniversity of Manchester 131 Princess Street Manchester M1 7DN U.K.

4. Mycobacterial Metabolism and Antibiotic Research LaboratoryThe Francis Crick Institute 1 Midland Road London NW1 1AT U.K.

5. Biomedical Sciences ProgramUniversity of Science and Technology Zewail City of Science and Technology Giza 12588 Egypt

6. Department of Chemistry College of Clinical PharmacyImam Abdulrahman Bin Faisal University Dammam Kingdom of Saudi Arabia

Funder

Biotechnology and Biological Sciences Research Council

Francis Crick Institute

Medical Research Council

Wellcome Trust

Diamond Light Source

Publisher

Wiley

Subject

General Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/open.201900227

Reference32 articles.

1. World Health Organization. Global tuberculosis report2017. Available from: http://www.who.int/tb/publications/global_report/en/ (accessed April 11 2019).

2. Drug-Resistant Tuberculosis

3. Advances in the development of new tuberculosis drugs and treatment regimens

4. Multidrug resistant tuberculosis

5. Structure, function and drug targeting in Mycobacterium tuberculosis cytochrome P450 systems

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