Design, Synthesis, Configuration Research, andIn VitroAntituberculosis Activities of two Chiral Naphthylamine Substituted Analogs of Bedaquiline-Reference-Cited by-同舟云学术

Design, Synthesis, Configuration Research, andIn VitroAntituberculosis Activities of two Chiral Naphthylamine Substituted Analogs of Bedaquiline

Published:2016-05-17 Issue:2 Volume:54 Page:1024-1030
ISSN:0022-152X
Container-title:Journal of Heterocyclic Chemistry
language:en
Short-container-title:J. Heterocyclic Chem.

Author:

Wang Zhiqiang¹²,Li Linwei¹,Zhou Zhixu¹,Geng Yiding¹,Chen Yu³,Sun Tiemin¹

Affiliation:

1. Key Laboratory of Structure-Based Drug Design and Discovery; Shenyang Pharmaceutical University, Ministry of Education; Shenyang 110016 People's Republic of China

2. College of Chemistry and Chemical Engineering; Harbin Normal University; Harbin 150025 People's Republic of China

3. School of Life Science and Biopharmaceutics; Shenyang Pharmaceutical University; Shenyang 110016 People's Republic of China

Publisher

Wiley

Subject

Organic Chemistry

Reference16 articles.

1. World Health Organization Tuberculosis Programme Global tuberculosis report 2013 http://www.who.int/tb/en/

2. A Diarylquinoline Drug Active on the ATP Synthase of Mycobacterium tuberculosis

3. Tucker , M. E. FDA Approves Bedaquiline for Resistant TB Treatment 2012

4. Design, Synthesis, and Pharmacological Evaluation of Mefloquine-Based Ligands as Novel Antituberculosis Agents

5. Synthesis, Crystal and Calculated Structure, and Biological Activity of 2-((6-Bromo-2-methoxyquinolin-3-yl) (phenyl)methyl)-2,3,7,7a-tetrahydro-3a,6-epoxyisoindol-1(6H)-one

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