Combating Multidrug‐Resistant Bacteria by Integrating a Novel Target Site Penetration and Receptor Binding Assay Platform Into Translational Modeling

Author:

Lang Yinzhi1,Shah Nirav R.1,Tao Xun1,Reeve Stephanie M.2,Zhou Jieqiang1,Moya Bartolome3,Sayed Alaa R. M.14,Dharuman Suresh2,Oyer Jeremiah L.5,Copik Alicja J.5,Fleischer Brett A.1,Shin Eunjeong1,Werkman Carolin1,Basso Kari B.6,Deveson Lucas Deanna7,Sutaria Dhruvitkumar S.1,Mégroz Marianne7,Kim Tae Hwan8,Loudon‐Hossler Victoria2,Wright Amy7,Jimenez‐Nieves Rossie H.1,Wallace Miranda J.2,Cadet Keisha C.1,Jiao Yuanyuan1,Boyce John D.7,LoVullo Eric D.9,Schweizer Herbert P.9,Bonomo Robert A.101112,Bharatham Nagakumar13,Tsuji Brian T.14,Landersdorfer Cornelia B.1516,Norris Michael H.17,Soo Shin Beom18,Louie Arnold19,Balasubramanian Venkataraman13,Lee Richard E.2,Drusano George L.19,Bulitta Jürgen B.1

Affiliation:

1. Department of Pharmacotherapy and Translational Research College of Pharmacy University of Florida Orlando Florida USA

2. Department of Chemical Biology and Therapeutics St. Jude Children’s Research Hospital Memphis Tennessee USA

3. Servicio de Microbiología and Unidad de Investigación Hospital Universitario Son Espases Instituto de Investigación Sanitaria Illes Balears (IdISBa) Palma de Mallorca Spain

4. Department of Chemistry Faculty of Science Fayoum University Fayoum Egypt

5. Burnett School of Biomedical Sciences College of Medicine University of Central Florida Orlando Florida USA

6. Department of Chemistry University of Florida Gainesville Florida USA

7. Infection and Immunity Program Department of Microbiology Monash Biomedicine Discovery Institute Monash University Melbourne Victoria Australia

8. College of Pharmacy Catholic University of Daegu Gyeongsan Gyeongbuk Korea

9. Pathogen and Microbiome Institute Northern Arizona University Flagstaff Arizona USA

10. Research Service and GRECC Louis Stokes Cleveland Department of Veterans Affairs Medical CenterCleveland Ohio USA

11. Department of Medicine, Pharmacology Molecular Biology and Microbiology Biochemistry and Proteomics and Bioinformatics Case Western Reserve University School of Medicine Cleveland Ohio USA

12. CWRU‐Cleveland VAMC Center for Antimicrobial Resistance and Epidemiology (Case VA CARES) Cleveland Ohio USA

13. BUGWORKS Research India Pvt. Ltd. Centre for Cellular & Molecular Platforms National Centre for Biological Sciences Bengaluru Karnataka India

14. Laboratory for Antimicrobial Pharmacodynamics University at Buffalo Buffalo New York USA

15. Drug Delivery, Disposition, and Dynamics Monash Institute of Pharmaceutical SciencesMonash University Melbourne Victoria Australia

16. Centre for Medicine Use and Safety Monash Institute of Pharmaceutical SciencesMonash University Melbourne Victoria Australia

17. Spatial Epidemiology and Ecology Research Laboratory Department of Geography and the Emerging Pathogens Institute University of Florida Gainesville Florida USA

18. School of Pharmacy Sungkyunkwan University Suwon Gyeonggi‐do Korea

19. Institute for Therapeutic Innovation College of Medicine University of Florida Orlando Florida USA

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Reference123 articles.

1. Clinical epidemiology of the global expansion of Klebsiella pneumoniae carbapenemases

2. Redfield R.R.CDC. Antibiotic resistant threats in the United States. Atlanta GA: U.S. Department of Health and Human Services US Centers for Disease Control and Prevention (2019) .

3. Looming Global-Scale Failures and Missing Institutions

4. Fix the antibiotics pipeline

5. Combating Antimicrobial Resistance: Policy Recommendations to Save Lives

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