Steric aspects of agonism and antagonism at β-adrenoceptors: Synthesis of and pharmacological experiments with the enantiomers of formoterol and their diastereomers-Reference-Cited by-同舟云学术

Steric aspects of agonism and antagonism at β-adrenoceptors: Synthesis of and pharmacological experiments with the enantiomers of formoterol and their diastereomers

Published:1991 Issue:6 Volume:3 Page:443-450
ISSN:0899-0042
Container-title:Chirality
language:en
Short-container-title:Chirality

Author:

Trofast Jan,ÖSterberg Kristina,Källström Britt-Louise,Waldeck Bertil

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Drug Discovery,Pharmacology,Catalysis,Analytical Chemistry

Reference27 articles.

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3. Absolute configuration of four isomers of 3-formamido-4-hydroxy-α-[[N-(p-methoxy-α-methylphenethyl)amino]methyl] benzylalcohol, a potent β-adrenoceptor stimulant;Murase;Chem. Pharm. Bull.,1978

4. Formoterol (AtockR): A new orally active and selective β2-receptor stimulant;Tasaka;Drugs Today,1986

5. The relation between biological activity and the degree of optical resolution of optical isomers;Barlow;J. Pharm. Pharmacol.,1972

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