Synthesis and pharmacological evaluation of fluorinated benzo[7]annulen-7-amines as GluN2B-selective NMDA receptor antagonists-Reference-Cited by-同舟云学术

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Synthesis and pharmacological evaluation of fluorinated benzo[7]annulen-7-amines as GluN2B-selective NMDA receptor antagonists

Published:2019-06-30 Issue:8 Volume:62 Page:354-379
ISSN:0362-4803
Container-title:Journal of Labelled Compounds and Radiopharmaceuticals
language:en
Short-container-title:J Label Compd Radiopharm

Author:

Thum Simone¹,Schepmann Dirk¹,Reinoso Raquel F.²,Alvarez Inés²,Ametamey Simon M.³^ORCID,Wünsch Bernhard¹⁴^ORCID

Affiliation:

1. Institute of Pharmaceutical and Medicinal Chemistry; Westfälische Wilhelms-Universität Münster; Münster Germany

2. Esteve Pharmaceuticals; Barcelona Spain

3. Center for Radiopharmaceutical Science of ETH, PSI, and USZ; ETH-Hönggerberg; Zürich Switzerland

4. Cells-in-Motion Cluster of Excellence (EXC 1003-CiM), Westfälische Wilhelms-Universität Münster; Germany

Funder

Deutsche Forschungsgemeinschaft

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Drug Discovery,Radiology Nuclear Medicine and imaging,Biochemistry,Analytical Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/jlcr.3718/fullpdf

Reference43 articles.

1. Crystal structure of a heterotetrameric NMDA receptor ion channel;Karakas;Science.,2014

2. A nomenclature for ligand-gated ion channels;Collingridge;Neuropharmacology.,2009

3. Funktion und potentielle therapeutische Bedeutung von NMDA-Rezeptoren. Teil 2: Therapiekonzepte und Rezeptorliganden;Stark;Pharm Unserer Zeit.,2000

4. Taming Glutamate excitotoxicity: strategic pathway modulation for neuroprotection;Jia;CNS Drugs.,2015

5. Allosteric modulators of NR2B-containing NMDA receptors: molecular mechanisms and therapeutic potential;Mony;Br J Pharmacol.,2009

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3. Conformationally Restricted σ₁ Receptor Antagonists from (−)-Isopulegol;Journal of Medicinal Chemistry;2023-03-22

4. Synthesis and biological evaluation of conformationally restricted GluN2B ligands derived from eliprodil;European Journal of Medicinal Chemistry;2022-07

5. A Review of Molecular Imaging of Glutamate Receptors;Molecules;2020-10-16

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