Single Stabilizing Point Mutation Enables High‐Resolution Co‐Crystal Structures of the Adenosine A <sub>2A</sub> Receptor with Preladenant Conjugates-Reference-Cited by-同舟云学术

Single Stabilizing Point Mutation Enables High‐Resolution Co‐Crystal Structures of the Adenosine A _2A Receptor with Preladenant Conjugates

Published:2022-03-24 Issue:22 Volume:61 Page:
ISSN:1433-7851
Container-title:Angewandte Chemie International Edition
language:en
Short-container-title:Angew Chem Int Ed

Author:

Claff Tobias¹^ORCID,Klapschinski Tim A.¹,Tiruttani Subhramanyam Udaya K.²³^ORCID,Vaaßen Victoria J.¹^ORCID,Schlegel Jonathan G.¹^ORCID,Vielmuth Christin¹,Voß Jan H.¹^ORCID,Labahn Jörg²³^ORCID,Müller Christa E.¹^ORCID

Affiliation:

1. Pharmaceutical Institute Pharmaceutical & Medicinal Chemistry University of Bonn An der Immenburg 4 53121 Bonn Germany

2. Centre for Structural Systems Biology (CSSB) Notkestraße 85 22607 Hamburg Germany

3. Research Centre Jülich Institute of Complex Systems (IBI-7) Wilhelm-Johnen-Straße 52425 Jülich Germany

Funder

Deutsche Forschungsgemeinschaft

Bundesministerium für Bildung und Forschung

Publisher

Wiley

Subject

General Chemistry,Catalysis

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/anie.202115545

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