TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics-Reference-Cited by-同舟云学术

TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics

Published:2020-07-15 Issue:46 Volume:59 Page:20338-20342
ISSN:1433-7851
Container-title:Angewandte Chemie International Edition
language:en
Short-container-title:Angew. Chem. Int. Ed.

Author:

Kunig Verena B. K.¹,Potowski Marco¹,Akbarzadeh Mohammad²,Klika Škopić Mateja¹,Santos Smith Denise¹,Arendt Lukas³,Dormuth Ina³,Adihou Hélène⁴⁵,Andlovic Blaž⁶⁷,Karatas Hacer²,Shaabani Shabnam⁸,Zarganes‐Tzitzikas Tryfon⁸,Neochoritis Constantinos G.⁸⁹,Zhang Ran⁸,Groves Matthew⁸,Guéret Stéphanie M.⁴⁵,Ottmann Christian⁷,Rahnenführer Jörg³,Fried Roland³,Dömling Alexander⁸,Brunschweiger Andreas¹^ORCID

Affiliation:

1. TU Dortmund University Faculty of Chemistry and Chemical Biology Otto-Hahn-Strasse 6 44227 Dortmund Germany

2. Max Planck Institute of Molecular Physiology Department of Chemical Biology Otto-Hahn-Strasse 11 44227 Dortmund Germany

3. TU Dortmund University Faculty of Statistics Vogelpothsweg 87 44227 Dortmund Germany

4. Medicinal Chemistry, Research and Early Development, Cardiovascular, Renal and Metabolism (CVRM) BioPharmaceuticals R&D AstraZeneca 43150 Gothenburg Sweden

5. AstraZeneca-Max Planck Institute Satellite Unit Max-Planck Institute of Molecular Physiology Department of Chemical Biology Otto-Hahn-Strasse 11 44227 Dortmund Germany

6. Lead Discovery Center GmbH (Germany) Otto-Hahn-Strasse 15 44227 Dortmund Germany

7. Laboratory of Chemical Biology Department of Biomedical Engineering and Institute for Complex Molecular Systems Eindhoven University of Technology Den Dolech 2 5612 AZ Eindhoven The Netherlands

8. University of Groningen Drug Design Deusinglaan 1 7313 AV Groningen The Netherlands

9. University of Crete Department of Chemistry 70013 Heraklion Greece

Funder

Deutsche Forschungsgemeinschaft

European Commission

National Institutes of Health

Hartstichting

Publisher

Wiley

Subject

General Chemistry,Catalysis

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