Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities-Reference-Cited by-同舟云学术

Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities

Published:2022-06-29 Issue:6 Volume:83 Page:1292-1304
ISSN:0272-4391
Container-title:Drug Development Research
language:en
Short-container-title:Drug Development Research

Author:

Keleş Atıcı Rüveyde¹,Doğan Şengül Dilem¹^ORCID,Gündüz Miyase Gözde²^ORCID,Krishna Vagolu Siva³,Chebaiki Melina⁴⁵,Homberset Håvard³,Lherbet Christian⁵,Mourey Lionel⁴,Tønjum Tone³⁶

Affiliation:

1. Department of Basic Sciences, Faculty of Pharmacy Erciyes University Kayseri Turkey

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy Hacettepe University Sıhhiye Ankara Turkey

3. Unit for Genome Dynamics, Department of Microbiology University of Oslo Oslo Norway

4. Institut de Pharmacologie et de Biologie Structurale, IPBS, Université de Toulouse, CNRS, UPS Toulouse France

5. LSPCMIB, UMR‐CNRS 5068, Université Paul Sabatier—Toulouse III Toulouse France

6. Unit for Genome Dynamics, Department of Microbiology Oslo University Hospital Oslo Norway

Publisher

Wiley

Subject

Drug Discovery

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ddr.21958

Reference44 articles.

1. Clickable conjugates of bile acids and nucleosides: Synthesis, characterization, in vitro anticancer and antituberculosis studies

2. Thiazole in the targeted anticancer drug discovery

3. Detection of katG and inhA mutations to guide isoniazid and ethionamide use for drug-resistant tuberculosis

4. The structure–activity relationship of urea derivatives as anti-tuberculosis agents

5. Drug discovery in tuberculosis. New drug targets and antimycobacterial agents

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