New Alkaloids and Steroids from Hydranth of Goniopora columna Corals and Their Inhibiting Lung Cancer Cell Activities

Author:

Feng Guangfu12ORCID,He Jieyi34,Li Qiqi12,Bai Meng12,Liu Kai12,Liu Xinming12,Yi Xiangxi2,Liu Yonghong12,Luo Lianxiang34,Gao Chenghai12ORCID

Affiliation:

1. Institute of Marine Drugs Guangxi University of Chinese Medicine Wuhe Road 13 530200 Nanning China

2. Guangxi Key Laboratory of Marine Drugs Guangxi University of Chinese Medicine Wuhe Road 13 530200 Nanning China

3. The Marine Biomedical Research Institute Guangdong Medical University Wenming East-Road 2 524023 Zhanjiang Guangdong China

4. The Marine Biomedical Research Institute of Guangdong Zhanjiang Wenming East-Road 2 524023 Zhanjiang Guangdong China

Abstract

AbstractA new alkaloids, aplysingoniopora A (1), and new configuration pregnane type steroid compound, 9,17‐α‐pregn‐1,4,20‐en‐3‐one (2), and two known pregnane type steroid compounds (3 and 4) were isolated from hydranth of Goniopora columna corals. The compounds structures and absolute configurations were determined by extensive spectroscopic analysis, MS data, single‐crystal X‐ray diffraction analysis and quantum chemical calculation. The anticancer effect of the compounds were explored in human non‐small‐cell lung cancer (NSCLC) A549 cell lines. As the results, the compound 3 and 4 induces toxicity and has proliferation inhibitory effects on A549 cells (IC50=58.99 μM and 58.77 μM, respectively) in vitro.

Funder

Guangdong Medical Research Foundation

Publisher

Wiley

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3