Thyrotropin receptor antagonists and inverse agonists, and their potential application to thyroid diseases
Author:
Affiliation:
1. Department of Molecular Medicine, Atomic Bomb Disease Institute, Nagasaki University, Nagasaki 852-8523, Japan
2. Center for Excellence in Thyroid Care, Kuma Hospital, Kobe 650-0011, Japan
Publisher
Japan Endocrine Society
Subject
Endocrinology,Endocrinology, Diabetes and Metabolism
Link
https://www.jstage.jst.go.jp/article/endocrj/69/11/69_EJ22-0391/_pdf
Reference58 articles.
1. 1 Davies TF, Andersen S, Latif R, Nagayama Y, Barbesino G, et al. (2020) Graves’ disease. Nat Rev Dis Primers 6: 52.
2. 2 Williams GR (2011) Extrathyroidal expression of TSH receptor. Ann Endocrinol (Paris) 72: 68–73.
3. 3 Rowe CW, Paul JW, Gedye C, Tolosa JM, Bendinelli C, et al. (2017) Targeting the TSH receptor in thyroid cancer. Endocr Relat Cancer 24: R191–R202.
4. 4 Kleinau G, Biebermann H (2014) Constitutive activities in the thyrotropin receptor: regulation and significance. Adv Pharmacol 70: 81–119.
5. 5 Vlaeminck-Guillem V, Ho SC, Rodien P, Vassart G, Costagliola S (2002) Activation of the cAMP pathway by the TSH receptor involves switching of the ectodomain from a tethered inverse agonist to an agonist. Mol Endocrinol 16: 736–746.
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