Thermal proteome profiling of breast cancer cells reveals proteasomal activation by CDK 4/6 inhibitor palbociclib

Author:

Miettinen Teemu P1234,Peltier Julien25,Härtlova Anetta25,Gierliński Marek6,Jansen Valerie M7,Trost Matthias25ORCID,Björklund Mikael1

Affiliation:

1. Division of Cell and Developmental Biology University of Dundee Dundee UK

2. MRC Protein Phosphorylation and Ubiquitylation Unit University of Dundee Dundee UK

3. MRC Laboratory for Molecular Cell Biology University College London London UK

4. Koch Institute for Integrative Cancer Research Massachusetts Institute of Technology Cambridge MA USA

5. Institute for Cell and Molecular Biosciences Newcastle University Newcastle upon Tyne UK

6. Division of Computational Biology University of Dundee Dundee UK

7. Division of Hematology‐Oncology Vanderbilt University Medical Center Nashville TN USA

Funder

AstraZeneca

Boehringer Ingelheim

GlaxoSmithKline

Janssen Pharmaceuticals

Merck KGaA

Pfizer

Wellcome Trust

Medical Research Council

Biotechnology and Biological Sciences Research Council

Conquer Cancer Foundation

Susan G. Komen

School of Medicine, Vanderbilt University

Publisher

EMBO

Subject

General Immunology and Microbiology,General Biochemistry, Genetics and Molecular Biology,Molecular Biology,General Neuroscience

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