Thio-β-D-glucosides: Synthesis and Evaluation as Glycosidase Inhibitors and Activators-Reference-Cited by-同舟云学术

Thio-β-D-glucosides: Synthesis and Evaluation as Glycosidase Inhibitors and Activators

Published:2014-08-21 Issue: Volume:2014 Page:1-8
ISSN:1687-9341
Container-title:International Journal of Carbohydrate Chemistry
language:en
Short-container-title:International Journal of Carbohydrate Chemistry

Author:

Samoshin Andrey V.¹,Dotsenko Irina A.¹,Samoshina Nataliya M.¹,Franz Andreas H.¹,Samoshin Vyacheslav V.¹

Affiliation:

1. Department of Chemistry, University of the Pacific, Stockton, CA 95211, USA

Abstract

Structurally simple 1-thio-β-D-glucopyranosides were synthesized and tested as potential inhibitors toward several fungal glycosidases from Aspergillus oryzae and Penicillium canescens. Significant selective inhibition was observed for α- and β-glucosidases, while a weak to moderate activation for α- and β-galactosidases.

Funder

National Science Foundation

Publisher

Hindawi Limited

Link

http://downloads.hindawi.com/archive/2014/941059.pdf

Reference52 articles.

1. Calixarene and Calixresorcarene Glycosides: Their Synthesis and Biological Applications

2. Synthesis and anti-inflammatory activity of aromatic glucosinolates

3. Aromatic thioglycoside inhibitors against the virulence factor LecA from Pseudomonas aeruginosa

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