Neurosteroid migration to intracellular compartments reduces steroid concentration in the membrane and diminishes GABA-A receptor potentiation
Author:
Publisher
Wiley
Subject
Physiology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1113/jphysiol.2007.142794/fullpdf
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3. Neuroactive steroids have multiple actions to potentiate GABAA receptors.;Akk;J Physiol,2004
4. Pregnenolone sulfate block of GABAA receptors: mechanism and involvement of a residue in the M2 region of the α subunit.;Akk;J Physiol,2001
5. Ethanol modulates the interaction of the endogenous neurosteroid allopregnanolone with the α1β2γ2L GABAA receptor.;Akk;Mol Pharmacol,2007
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