AMG 176, a Selective MCL1 Inhibitor, is Effective in Hematological Cancer Models Alone and in Combination with Established Therapies

Author:

Caenepeel Sean,Brown Sean PORCID,Belmontes Brian,Moody Gordon,Keegan Kathleen S,Chui Danny,Whittington Douglas A.,Huang Xin,Poppe Leszek,Cheng Alan C.,Cardozo Mario,Houze Jonathan,Li Yunxiao,Lucas Brian,Paras Nick A.ORCID,Wang Xianghong,Taygerly Joshua P,Vimolratana Marc,Zancanella Manuel,Zhu Liusheng,Cajulis Elaina,Osgood Tao,Sun Jan,Damon LeahORCID,Egan Regina K.,Greninger PatriciaORCID,McClanaghan Joseph D,Gong Jianan,Moujalled Donia,Pomilio Giovanna,Beltran Pedro,Benes Cyril H.ORCID,Roberts Andrew W.ORCID,Huang David C.S.ORCID,Wei Andrew,Canon Jude,Coxon Angela,Hughes Paul E.

Funder

Amgen (Amgen Inc.)

Australian Cancer Research Foundation (ACRF)

Department of Health | National Health and Medical Research Council (NHMRC)

Independent Research Institutes

The Cancer Council Victoria

Leukemia and Lymphoma Society (LLS)

Publisher

American Association for Cancer Research (AACR)

Subject

Oncology

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