Quantifying the CDK inhibitor VMY-1-103’s activity and tissue levels in an in vivo tumor model by LC-MS/MS and by MRI

Author:

Sirajuddin Paul1,Das Sudeep2,Ringer Lymor1,Rodriguez Olga C.1,Sivakumar Angiela1,Lee Yi-Chien1,Uren Aykut1,Fricke Stanley T.3,Rood Brian3,Ozcan Alpay4,Wang Sean S.1,Karam Sana5,Yenugonda Venkata6,Salinas Patricia1,Petricoin III Emanuel7,Pishvaian Michael1,Lisanti Michael P.8,Wang Yue49,Schlegel Richard110,Moasser Bahram2,Albanese Chris110

Affiliation:

1. Lombardi Comprehensive Cancer Center and Department of Oncology; Georgetown University Medical Center; Washington, DC USA

2. Department of Chemistry; Georgetown University; Washington, DC USA

3. Children’s National Medical Center; Washington, DC USA

4. Department of Physics; Virginia Tech; Arlington, VA USA

5. Department of Radiation Biology; Georgetown University Medical Center; Washington, DC USA

6. Drug Discovery Program; Georgetown University Medical Center; Washington, DC USA

7. Center for Applied Proteomics and Molecular Medicine; School of Systems Biology; George Mason University; Manassas, VA USA

8. Department Stem Cell Biology; Kimmel Cancer Center; Thomas Jefferson University; Philadelphia, PA USA

9. Bradley Department of Electrical and Computer Engineering; Virginia Tech; Arlington, VA USA

10. Department of Pathology; Georgetown University Medical Center; Washington, DC USA

Publisher

Informa UK Limited

Subject

Cell Biology,Developmental Biology,Molecular Biology

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