Evaluation of the alpha 2-adrenoceptor blocking properties of buspirone and ipsapirone in healthy subjects. Relationship with the plasma concentration of the common metabolite 1-(2-pyrimidinyl)-piperazine.-Reference-Cited by-同舟云学术

Evaluation of the alpha 2-adrenoceptor blocking properties of buspirone and ipsapirone in healthy subjects. Relationship with the plasma concentration of the common metabolite 1-(2-pyrimidinyl)-piperazine.

Published:1995-03 Issue:3 Volume:39 Page:243-249
ISSN:0306-5251
Container-title:British Journal of Clinical Pharmacology
language:en
Short-container-title:British Journal of Clinical Pharmacology

Author:

Berlin I,Chalon S,Payan C,Schollnhammer G,Cesselin F,Varoquaux O,Puech AJ

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1365-2125.1995.tb04443.x/fullpdf

Reference35 articles.

1. 1-(2-Pyrimidinyl)-piperazine may alter the effects of the 5HT1A agonists in the learned helplessness paradigm in rats;Martin;Psychopharmacology,1991

2. Reversal of helpless behaviour in rats by putative 5-HT1A agonists;Giral;Biol Psychiatry,1988

3. 1-(2-pyrimidinyl)-piperazine as active metabolite of buspirone in man and rat;Caccia;Pharmacology,1986

4. Blockade of α2-adrenoceptors by 1-(-pyrimidinyl)-piperazine (PmP) in vivo and its relation to the activity of buspirone;Bianchi;Eur J Pharmac,1988

5. The α2-adrenoceptor antagonist activity of ipsapirone and gepirone is mediated by their common metabolite 1-(2-pyrimidinyl)-piperazine (PmP);Bianchi;Eur J Pharmac,1988

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