Synthesis and evaluation of C3 substituted chalcone‐based derivatives of 7‐azaindole as protein kinase inhibitors-Reference-Cited by-同舟云学术

Synthesis and evaluation of C3 substituted chalcone‐based derivatives of 7‐azaindole as protein kinase inhibitors

Published:2020-08-18 Issue:6 Volume:96 Page:1395-1407
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Qhobosheane Malikotsi A.¹^ORCID,Legoabe Lesetja J.¹^ORCID,Josselin Béatrice²³,Bach Stéphane²³,Ruchaud Sandrine²,Beteck Richard M.¹^ORCID

Affiliation:

1. Centre of Excellence for Pharmaceutical Sciences North‐West University Potchefstroom South Africa

2. Sorbonne Université CNRS UMR 8227 Integrative Biology of Marine Models Laboratory (LBI2M) Station Biologique de Roscoff Roscoff Cedex France

3. Sorbonne Université CNRS FR2424 Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening facility) Station Biologique de Roscoff Roscoff France

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.13748

Reference27 articles.

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5. Progress towards a public chemogenomic set for protein kinases and a call for contributions

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1. Assessment of Polyphenol Oxidase Inhibition, Antimicrobial and Antioxidant Properties of Some Chalcone Derivates: Experimental and Computational Approaches;2024

2. Laser spectroscopic characterization of supersonic jet cooled 2,7-diazaindole;Physical Chemistry Chemical Physics;2023

3. Function and inhibition of Haspin kinase: targeting multiple cancer therapies by antimitosis;Journal of Pharmacy and Pharmacology;2022-11-05

4. Exploration of 7-azaindole-coumaranone hybrids and their analogues as protein kinase inhibitors;Chemico-Biological Interactions;2021-07