Research Letter: Structural Combination of Established 5-HT2A Receptor Ligands: New Aspects of the Binding Mode-Reference-Cited by-同舟云学术

Research Letter: Structural Combination of Established 5-HT2A Receptor Ligands: New Aspects of the Binding Mode

Published:2010-07-15 Issue:4 Volume:76 Page:361-366
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:

Author:

Kramer Vasko,Herth Matthias M.,Santini Martin A.,Palner Mikael,Knudsen Gitte M.,Rösch Frank

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Reference17 articles.

1. Development of a Receptor-Interaction Model for Serotonin 5-HT2A Receptor Antagonists. Predicting Selectivity with Respect to Dopamin D2 Receptors;Andersen;J Med Chem,1994

2. Classification of typical and atypical antipsychotic drugs on the basis of dopamin D-1, D-2 and serotonin2 pKi values;Meltzer;J Pharmacol Exp Ther,1989

3. Enhanced 5-HT2A receptor status in the hypothalamus and corpus striatum of ethanol-treated rats;Akash;Cell Mol Neurobiol,2008

4. Reduced 5-HT2A receptor binding in patients with mild cognitive impairment;Hasselbalch;Neurobiol Aging,2008

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The Benzoylpiperidine Fragment as a Privileged Structure in Medicinal Chemistry: A Comprehensive Review;Molecules;2024-04-23

2. Serotonin2B receptor blockade in the rat dorsal raphe nucleus suppresses cocaine-induced hyperlocomotion through an opposite control of mesocortical and mesoaccumbens dopamine pathways;Neuropharmacology;2020-12

3. Serotonin2B receptors in the rat dorsal raphe nucleus exert a GABA-mediated tonic inhibitory control on serotonin neurons;Experimental Neurology;2019-01

4. PET Imaging of the 5-HT2A Receptor System: A Tool to Study the Receptor’s In Vivo Brain Function;5-HT2A Receptors in the Central Nervous System;2018

5. Current radiosynthesis strategies for 5-HT2Areceptor PET tracers;Journal of Labelled Compounds and Radiopharmaceuticals;2015-05-22