PKPD modelling to predict altered disposition of 1α,25-dihydroxyvitamin D3in mice due to dose-dependent regulation of CYP27B1 on synthesis and CYP24A1 on degradation
Author:
Affiliation:
1. Department of Pharmaceutical Sciences, Leslie Dan Faculty of Pharmacy; University of Toronto; Toronto Ontario Canada
2. Department of Pharmaceutical Sciences, University at Buffalo; State University of New York; Buffalo NY USA
Funder
CIHR
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/bph.13153/fullpdf
Reference50 articles.
1. Induction of vitamin D 24-hydroxylase messenger RNA and activity by 22-oxacalcitriol in mouse kidney and duodenum. Possible role in decrease of plasma 1α,25-dihydroxyvitamin D3;Akeno;Biochem Pharmacol,1994
2. The Concise Guide to PHARMACOLOGY 2013/14: ion channels;Alexander;Br J Pharmacol,2013a
3. The Concise Guide to PHARMACOLOGY 2013/14: nuclear hormone receptors;Alexander;Br J Pharmacol,2013b
4. The Concise Guide to PHARMACOLOGY 2013/14: enzymes;Alexander;Br J Pharmacol,2013c
5. Statistical estimations in pharmacokinetics;Boxenbaum;J Pharmacokinet Biopharm,1974
Cited by 6 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Physiologically Based Pharmacokinetic Modeling of Vitamin D3 and Metabolites in Vitamin D–Insufficient Patients;Drug Metabolism and Disposition;2022-07-02
2. Noteworthy idiosyncrasies of 1α,25‐dihydroxyvitamin D3kinetics for extrapolation from mouse to man: Commentary;Biopharmaceutics & Drug Disposition;2020-03
3. Involvement of RBP4 in Diabetic Atherosclerosis and the Role of Vitamin D Intervention;Journal of Diabetes Research;2018-08-16
4. Potencies of vitamin D analogs, 1α-hydroxyvitamin D3 , 1α-hydroxyvitamin D2 and 25-hydroxyvitamin D3 , in lowering cholesterol in hypercholesterolemic mice in vivo;Biopharmaceutics & Drug Disposition;2018-04
5. Highlighting Vitamin D Receptor–Targeted Activities of 1α,25-Dihydroxyvitamin D3in Mice via Physiologically Based Pharmacokinetic-Pharmacodynamic Modeling;Drug Metabolism and Disposition;2017-10-30
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3